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Search Results for " adrenoceptor antagonist "

20

Compounds

Cat No. Product Name Synonyms Targets
T22033 ARC 239 dihydrochloride Norepinephrine
ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).
T23301 (S)-(+)-Niguldipine hydrochloride Others
(S)-(+)-Niguldipine hydrochloride is a L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist.
T12597 5-HT2 antagonist 1 5-HT Receptor
5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.
T26923 Bunazosin Hydrochloride E 1015,E643,E-1015,E-643,E 643 Adrenergic Receptor
Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.
T30027 Amosulalol Adrenergic Receptor
Amosulalol is a combined alpha and beta adrenoceptor antagonist.
T28922 Taprizosin Taprizosin Mesylate,UK-338003,UK-338,003,UK338003,UK 338003 Adrenergic Receptor
Taprizosin(UK-338003) is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.
T61535 Neldazosin Adrenergic Receptor
Neldazosin is used as a potent α1-adrenoceptor antagonist.
T28267 ORM-10921 ORM10921,ORM 10921 Adrenergic Receptor
ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.
T11726 JP1302 dihydrochloride Adrenergic Receptor
JP1302 dihydrochloride is a selective, high affinity antagonist of the alpha2C-adrenoceptor (α2C-adrenoceptor), with a Ki (binding affinity) value of 28 nM and a Kb value (antagonist activity) of 16 nM.
T30846 CGP-20712 UNII-SIO2UEZ19H,CGP 20712 Adrenergic Receptor
CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.
T35326 Labetalone hydrochloride Labetalone hydrochloride,Benzoic amide Others
Labetalone hydrochloride (Benzoic amide) is an impurity of Labetalol. Labetalol is an orally active adrenoceptor blocking drug, Labetalol is a competitive antagonist at both alpha- and beta-adrenoceptor sites
T10812 Cicloprolol hydrochloride Adrenergic Receptor
Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.
T11286 Fiduxosin A 185980.1,ABT 980 Adrenergic Receptor
Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with Ki values of 0.160 nM, 24.9 nM and 0.920 nM, respectively. Fiduxosin...
T16431 Pamatolol Adrenergic Receptor
Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments.
T11015 Midaglizole hydrochloride (±)-DG5128,(±)-DG5128 hydrochloride,DG5128 hydrochloride,DG5128 Adrenergic Receptor
Midaglizole hydrochloride ((±)-DG5128) (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenoceptor (pKi = 6.28) 7.4 times higher than that of α1-adrenocepto...
T0088 Urapidil hydrochloride Urapidil HCl 5-HT Receptor , Adrenergic Receptor
Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
T9220 Naftopidil hydrochloride 1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-,KT-611 hydrochloride,BM-15275 hydrochloride Adrenergic Receptor
Naftopidil hydrochloride (BM-15275 hydrochloride) is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, respective...
T20898 (R)-Propranolol hydrochloride Dexpropranolol hydrochloride,(R)-(+)-Propranolol Adrenergic Receptor
(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol. Propranolol is a nonselective β-adrenergic receptor (βAR) antag...
T7079 Batefenterol GSK961081,TD-5959 Adrenergic Receptor , AChR
Batefenterol (TD-5959) (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor (Ki:1.4/1.3/3.7 nM).
T12643 (R)-Terazosin Adrenergic Receptor
(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values of 6.51 nM, 1.01 nM and 1.97 nM, respectively).

Compounds

ARC 239 dihydrochloride
T22033
Synonym:
Target: Norepinephrine
(S)-(+)-Niguldipine hydrochloride
T23301
Synonym:
Target: Others
5-HT2 antagonist 1
T12597
Synonym:
Target: 5-HT Receptor
Bunazosin Hydrochloride
T26923
Synonym: E 1015,E643,E-1015,E-643,E 643
Target: Adrenergic Receptor
Amosulalol
T30027
Synonym:
Target: Adrenergic Receptor
Taprizosin
T28922
Synonym: Taprizosin Mesylate,UK-338003,UK-338,003,UK338003,UK 338003
Target: Adrenergic Receptor
Neldazosin
T61535
Synonym:
Target: Adrenergic Receptor
ORM-10921
T28267
Synonym: ORM10921,ORM 10921
Target: Adrenergic Receptor
JP1302 dihydrochloride
T11726
Synonym:
Target: Adrenergic Receptor
CGP-20712
T30846
Synonym: UNII-SIO2UEZ19H,CGP 20712
Target: Adrenergic Receptor
Labetalone hydrochloride
T35326
Synonym: Labetalone hydrochloride,Benzoic amide
Target: Others
Cicloprolol hydrochloride
T10812
Synonym:
Target: Adrenergic Receptor
Fiduxosin
T11286
Synonym: A 185980.1,ABT 980
Target: Adrenergic Receptor
Pamatolol
T16431
Synonym:
Target: Adrenergic Receptor
Midaglizole hydrochloride
T11015
Synonym: (±)-DG5128,(±)-DG5128 hydrochloride,DG5128 hydrochloride,DG5128
Target: Adrenergic Receptor
Urapidil hydrochloride
T0088
Synonym: Urapidil HCl
Target: 5-HT Receptor, Adrenergic Receptor
Naftopidil hydrochloride
T9220
Synonym: 1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-,KT-611 hydrochloride,BM-15275 hydrochloride
Target: Adrenergic Receptor
(R)-Propranolol hydrochloride
T20898
Synonym: Dexpropranolol hydrochloride,(R)-(+)-Propranolol
Target: Adrenergic Receptor
Batefenterol
T7079
Synonym: GSK961081,TD-5959
Target: Adrenergic Receptor, AChR
(R)-Terazosin
T12643
Synonym:
Target: Adrenergic Receptor
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TargetMol