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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T22033 | ARC 239 dihydrochloride | Norepinephrine | |
ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively). | |||
T23301 | (S)-(+)-Niguldipine hydrochloride | Others | |
(S)-(+)-Niguldipine hydrochloride is a L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist. | |||
T12597 | 5-HT2 antagonist 1 | 5-HT Receptor | |
5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity. | |||
T26923 | Bunazosin Hydrochloride | E 1015,E643,E-1015,E-643,E 643 | Adrenergic Receptor |
Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug. | |||
T30027 | Amosulalol | Adrenergic Receptor | |
Amosulalol is a combined alpha and beta adrenoceptor antagonist. | |||
T28922 | Taprizosin | Taprizosin Mesylate,UK-338003,UK-338,003,UK338003,UK 338003 | Adrenergic Receptor |
Taprizosin(UK-338003) is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia. | |||
T61535 | Neldazosin | Adrenergic Receptor | |
Neldazosin is used as a potent α1-adrenoceptor antagonist. | |||
T28267 | ORM-10921 | ORM10921,ORM 10921 | Adrenergic Receptor |
ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies. | |||
T11726 | JP1302 dihydrochloride | Adrenergic Receptor | |
JP1302 dihydrochloride is a selective, high affinity antagonist of the alpha2C-adrenoceptor (α2C-adrenoceptor), with a Ki (binding affinity) value of 28 nM and a Kb value (antagonist activity) of 16 nM. | |||
T30846 | CGP-20712 | UNII-SIO2UEZ19H,CGP 20712 | Adrenergic Receptor |
CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM. | |||
T35326 | Labetalone hydrochloride | Labetalone hydrochloride,Benzoic amide | Others |
Labetalone hydrochloride (Benzoic amide) is an impurity of Labetalol. Labetalol is an orally active adrenoceptor blocking drug, Labetalol is a competitive antagonist at both alpha- and beta-adrenoceptor sites | |||
T10812 | Cicloprolol hydrochloride | Adrenergic Receptor | |
Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease. | |||
T11286 | Fiduxosin | A 185980.1,ABT 980 | Adrenergic Receptor |
Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with Ki values of 0.160 nM, 24.9 nM and 0.920 nM, respectively. Fiduxosin... | |||
T16431 | Pamatolol | Adrenergic Receptor | |
Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments. | |||
T11015 | Midaglizole hydrochloride | (±)-DG5128,(±)-DG5128 hydrochloride,DG5128 hydrochloride,DG5128 | Adrenergic Receptor |
Midaglizole hydrochloride ((±)-DG5128) (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenoceptor (pKi = 6.28) 7.4 times higher than that of α1-adrenocepto... | |||
T0088 | Urapidil hydrochloride | Urapidil HCl | 5-HT Receptor , Adrenergic Receptor |
Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist. | |||
T9220 | Naftopidil hydrochloride | 1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-,KT-611 hydrochloride,BM-15275 hydrochloride | Adrenergic Receptor |
Naftopidil hydrochloride (BM-15275 hydrochloride) is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, respective... | |||
T20898 | (R)-Propranolol hydrochloride | Dexpropranolol hydrochloride,(R)-(+)-Propranolol | Adrenergic Receptor |
(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol. Propranolol is a nonselective β-adrenergic receptor (βAR) antag... | |||
T7079 | Batefenterol | GSK961081,TD-5959 | Adrenergic Receptor , AChR |
Batefenterol (TD-5959) (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor (Ki:1.4/1.3/3.7 nM). | |||
T12643 | (R)-Terazosin | Adrenergic Receptor | |
(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values of 6.51 nM, 1.01 nM and 1.97 nM, respectively). |